a 301 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T33725	Norgestrienone	Planor,A-301,A301,Ogyline,A 301
	Nogotrienone is an anabolic steroid with fertility and contraceptive activity that has been studied as a therapeutic agent for hereditary angioneurotic edema.
T7425	RU-301		TAM Receptor
	RU-301 is a novel pan-tam inhibitor		TAM Receptor
T9212	IMB-301		Others , HIV Protease
	IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.		Others , HIV Protease
T29021	TT-301	MW 189,MW189,TT301,TT 301,MW 189 ;MW189,MW-189
	TT-301 is a cytokine inhibitor and glial cell inhibitor.
T28423	PKUMDL-LTQ-301
	PKUMDL-LTQ-301 is a potent inhibitor of HipA toxin. PKUMDL-LTQ-301 also inhibits E. coli persistence.
T71077	UH 301
	UH 301 is a 5-HT1A receptor antagonist.
T17095	TIK-301	PD-6735,LY-156735	5-HT Receptor
	TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM, respectively). TIK-301 is also a 5-HT2B/5-HT2C receptor an...		5-HT Receptor
T73458	LWG-301
	LWG-301, an allosteric inhibitor of Glutaminase 1 (GLS1), demonstrates a potent inhibition with an IC50 value of 7 nM. It effectively impedes glutamine metabolism and elevates intracellular ROS levels, thereby inducing a...
T34958	TRK-380	TAC301,TAC 301,TAC-301,TRK 380,TRK380
	TRK-380 (TAC-301) is an effective and selective β3-adrenergic receptor agonist. TRK-380 improves formalin-induced frequent urination in rats and carbachol-induced bladder contraction in dogs (a decrease of 37.6%).
T76949	Zelminemab
	Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].
T69577	LEI-301
	LEI-301 is a novel potent inhibitor for the PLAAT family members, reducing the NAE levels, including anandamide, in cells overexpressing PLAAT2 or PLAAT5.
T73156	LabMol-301
	LabMol-301, a chemical compound, effectively inhibits NS5 RdRp and NS2B-NS3pro activity with IC50 values of 0.8 μM and 7.4 μM, respectively. Additionally, it exhibits cytoprotective effects, safeguarding against Zika vir...
T81554	Pancreastatin (37-52), human
	Pancreastatin (37-52), human, is a biologically active fragment of CgA-derived peptide (residues 250–301) that inhibits insulin release from islet beta cells [1][2].
T80494	Tap1a	TRTX-Tap1a,Theraphotoxin-Tap1a,µ/ω-TRTX-Tap1a	Sodium Channel
	Theraphotoxin-Tap1a (Tap1a) is a spider venom-derived peptide that acts as an inhibitor of sodium channels, displaying IC50 values of 80 nM for Na v 1.7 and 301 nM for Na v 1.1. It demonstrates analgesic effects [1].		Sodium Channel
T81708	Nagrestipen
	Nagrestipen, a variant of the human macrophage inflammatory protein-1 alpha (MIP-1α), also referred to as ECI 301, exhibits antitumor activity. It is employed in therapeutic trials focused on cancer, assessing its effica...
T83328	4A7C-301
	4A7C-301, a Nurr1 agonist, exhibits potent neuroprotective effects in vitro and markedly mitigates neuropathological abnormalities while enhancing motor and olfactory functions in male mouse models with AAV2-mediated α-s...
T77151	Cosibelimab
	Cosibelimab (CK-301; TG-1501) is a fully human, high-affinity monoclonal antibody that inhibits PD-L1 by preventing its interaction with PD-1. This compound, featuring a functional Fc domain, is effective in inducing ant...
T83894	4A7C-301-Nurr1 Agonist	4A7C-301-Nuclear Receptor-Related 1
	The compound 4A7C-301-Nurr1 agonist is a specific agonist for the nuclear receptor-related 1 (Nurr1). By binding to the Nurr1 ligand-binding domain with an IC50 value of 48.22 nM, it enhances the transcriptional activity...
T62090	(Rac)-Tanomastat
	Rac)-Tanomastat ((Rac)-BAY 12-9566) is a racemate of Tanomastat. Tanomastat (BAY 12-9566) is an orally active, zinc carboxy-containing inhibitor of non-peptide biphenyl matrix metalloproteinases (MMPs) that inhibits MMP-...
T76973	Tosatoxumab
	Tosatoxumab (AR-301; KBSA301), a human immunoglobulin G1 monoclonal antibody, specifically targets and neutralizes S. aureus alpha-toxin (alpha-hemolysin; Hla) by binding to its N-terminal epitope. This interaction block...